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Exploring the epige...
Exploring the epigenetic drug discovery landscape
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- Prachayasittikul, Veda (författare)
- Mahidol Univ, Fac Med Technol, Ctr Data Min & Biomed Informat, Bangkok, Thailand.
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- Prathipati, Philip (författare)
- Natl Inst Biomed Innovat, Osaka, Japan.;Natl Inst Hlth & Nutr, Osaka, Japan.
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- Pratiwi, Reny (författare)
- Mahidol Univ, Fac Med Technol, Ctr Data Min & Biomed Informat, Bangkok, Thailand.
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- Phanus-umporn, Chuleeporn (författare)
- Mahidol Univ, Fac Med Technol, Ctr Data Min & Biomed Informat, Bangkok, Thailand.
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- Malik, Aijaz Ahmad (författare)
- Mahidol Univ, Fac Med Technol, Ctr Data Min & Biomed Informat, Bangkok, Thailand.
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- Schaduangrat, Nalini (författare)
- Mahidol Univ, Fac Med Technol, Ctr Data Min & Biomed Informat, Bangkok, Thailand.
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- Seenprachawong, Kanokwan (författare)
- Mahidol Univ, Fac Med Technol, Dept Clin Microscopy, Bangkok, Thailand.
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- Wongchitrat, Prapimpun (författare)
- Mahidol Univ, Fac Med Technol, Ctr Res & Innovat, Bangkok, Thailand.
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- Supokawej, Aungkura (författare)
- Mahidol Univ, Fac Med Technol, Dept Clin Microscopy, Bangkok, Thailand.
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- Prachayasittikul, Virapong (författare)
- Mahidol Univ, Fac Med Technol, Dept Clin Microbiol & Appl Technol, Bangkok, Thailand.
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- Wikberg, Jarl E. S. (författare)
- Uppsala universitet,Institutionen för farmaceutisk biovetenskap
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- Nantasenamat, Chanin (författare)
- Mahidol Univ, Fac Med Technol, Ctr Data Min & Biomed Informat, Bangkok, Thailand.
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Mahidol Univ, Fac Med Technol, Ctr Data Min & Biomed Informat, Bangkok, Thailand Natl Inst Biomed Innovat, Osaka, Japan.;Natl Inst Hlth & Nutr, Osaka, Japan. (creator_code:org_t)
- 2017-02-28
- 2017
- Engelska.
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Ingår i: Expert Opinion on Drug Discovery. - : TAYLOR & FRANCIS LTD. - 1746-0441 .- 1746-045X. ; 12:4, s. 345-362
- Relaterad länk:
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https://urn.kb.se/re...
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https://doi.org/10.1...
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Abstract
Ämnesord
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- Introduction: Epigenetic modification has been implicated in a wide range of diseases and the ability to modulate such systems is a lucrative therapeutic strategy in drug discovery. Areas covered: This article focuses on the concepts and drug discovery aspects of epigenomics. This is achieved by providing a survey of the following concepts: (i) factors influencing epigenetics, (ii) diseases arising from epigenetics, (iii) epigenetic enzymes as druggable targets along with coverage of existing FDA-approved drugs and pharmacological agents, and (iv) drug repurposing/repositioning as a means for rapid discovery of pharmacological agents targeting epigenetics. Expert opinion: Despite significant interests in targeting epigenetic modifiers as a therapeutic route, certain classes of target proteins are heavily studied while some are less characterized. Thus, such orphan target proteins are not yet druggable with limited report of active modulators. Current research points towards a great future with novel drugs directed to the many complex multifactorial diseases of humans, which are still often poorly understood and difficult to treat.
Ämnesord
- MEDICIN OCH HÄLSOVETENSKAP -- Medicinska och farmaceutiska grundvetenskaper -- Farmakologi och toxikologi (hsv//swe)
- MEDICAL AND HEALTH SCIENCES -- Basic Medicine -- Pharmacology and Toxicology (hsv//eng)
Nyckelord
- Epigenomics
- epigenetics
- drug discovery
- drugs
- bioinformatics
- cheminformatics
- chemogenomics
- proteochemometrics
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