Search: onr:"swepub:oai:DiVA.org:umu-32675" >
Improved procedure ...
Improved procedure for the enantioselective synthesis of dihydrooxazolo and dihydrothiazolo ring-fused 2-pyridones
-
- Chorell, Erik, 1980- (author)
- Umeå universitet,Kemiska institutionen,Fredrik Almqvist
-
- Edvinsson, Sofie (author)
- Umeå universitet,Kemiska institutionen
-
- Almqvist, Fredrik (author)
- Umeå universitet,Kemiska institutionen
-
(creator_code:org_t)
- Elsevier Ltd, 2010
- 2010
- English.
-
In: Tetrahedron Letters. - : Elsevier Ltd. - 0040-4039 .- 1359-8562. ; 51:18, s. 2461-2463
- Related links:
-
https://urn.kb.se/re...
-
show more...
-
https://doi.org/10.1...
-
show less...
Abstract
Subject headings
Close
- Improved procedures to synthesize enantioselectively analogues of a peptidomimetic scaffold with high biological relevance have been developed. Experimental design led to a general method for the preparation of dihydrooxazolo ring-fused 2-pyridones in good yields and high enantiomeric purity. The knowledge gained from this was also used to improve the microwave-accelerated synthesis of dihydrothiazolo ring-fused 2-pyridones to give complete stereo retention and high yields.
Keyword
- 2-Pyridone
- PPTS
- Peptidomimetic
- Enantioselective
- Pilicide
- Curlicide
Publication and Content Type
- ref (subject category)
- art (subject category)
Find in a library
To the university's database