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Flavonoids as dual-...
Flavonoids as dual-target inhibitors against α-glucosidase and α-amylase : a systematic review of in vitro studies
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- Lam, Thua-Phong (författare)
- Uppsala universitet,Institutionen för farmaci,Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.
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- Tran, Ngoc-Vi Nguyen (författare)
- Uppsala universitet,Institutionen för farmaci,Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.
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- Pham, Long-Hung Dinh (författare)
- Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.;Imperial Coll London, Dept Chem, London W12 0BZ, England.
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- Lai, Nghia Vo-Trong (författare)
- Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.
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- Dang, Bao-Tran Ngoc (författare)
- Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.
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- Truong, Ngoc-Lam Nguyen (författare)
- Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.
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- Nguyen-Vo, Song-Ky (författare)
- Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.
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- Hoang, Thuy-Linh (författare)
- Calif Northstate Univ, Coll Pharm, Elk Grove, CA 95757 USA.
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- Mai, Tan Thanh (författare)
- Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.
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- Tran, Thanh-Dao (författare)
- Univ Med & Pharm Ho Chi Minh City, Fac Pharm, Ho Chi Minh City 700000, Vietnam.
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(creator_code:org_t)
- Springer, 2024
- 2024
- Engelska.
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Ingår i: NATURAL PRODUCTS AND BIOPROSPECTING. - : Springer. - 2192-2195 .- 2192-2209. ; 14:1
- Relaterad länk:
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https://doi.org/10.1...
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https://uu.diva-port... (primary) (Raw object)
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https://urn.kb.se/re...
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https://doi.org/10.1...
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Abstract
Ämnesord
Stäng
- Diabetes mellitus remains a major global health issue, and great attention is directed at natural therapeutics. This systematic review aimed to assess the potential of flavonoids as antidiabetic agents by investigating their inhibitory effects on alpha-glucosidase and alpha-amylase, two key enzymes involved in starch digestion. Six scientific databases (PubMed, Virtual Health Library, EMBASE, SCOPUS, Web of Science, and WHO Global Index Medicus) were searched until August 21, 2022, for in vitro studies reporting IC50 values of purified flavonoids on alpha-amylase and alpha-glucosidase, along with corresponding data for acarbose as a positive control. A total of 339 eligible articles were analyzed, resulting in the retrieval of 1643 flavonoid structures. These structures were rigorously standardized and curated, yielding 974 unique compounds, among which 177 flavonoids exhibited inhibition of both alpha-glucosidase and alpha-amylase are presented. Quality assessment utilizing a modified CONSORT checklist and structure-activity relationship (SAR) analysis were performed, revealing crucial features for the simultaneous inhibition of flavonoids against both enzymes. Moreover, the review also addressed several limitations in the current research landscape and proposed potential solutions. The curated datasets are available online at https://github.com/MedChemUMP/FDIGA.
Ämnesord
- LANTBRUKSVETENSKAPER -- Lantbruksvetenskap, skogsbruk och fiske -- Livsmedelsvetenskap (hsv//swe)
- AGRICULTURAL SCIENCES -- Agriculture, Forestry and Fisheries -- Food Science (hsv//eng)
Nyckelord
- Systematic review
- Flavonoids
- Dual-target
- Glucosidase
- Amylase
- PRISMA
- SAR
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Lam, Thua-Phong
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Tran, Ngoc-Vi Ng ...
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Pham, Long-Hung ...
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Lai, Nghia Vo-Tr ...
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Dang, Bao-Tran N ...
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Truong, Ngoc-Lam ...
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Nguyen-Vo, Song- ...
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Hoang, Thuy-Linh
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Mai, Tan Thanh
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Tran, Thanh-Dao
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