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024 | 7 | a https://gup.ub.gu.se/publication/3344322 URI |
024 | 7 | a https://doi.org/10.1111/bph.161772 DOI |
024 | 7 | a https://urn.kb.se/resolve?urn=urn:nbn:se:uu:diva-5218952 URI |
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100 | 1 | a Alexander, Stephen P. H.u Univ Nottingham, Med Sch, Sch Life Sci, Nottingham NG7 2UH, England.4 aut |
245 | 1 0 | a The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors |
264 | 1 | b British pharmacological society,c 2023 |
520 | a The Concise Guide to PHARMACOLOGY 2023/24 is the sixth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of approximately 1800 drug targets, and about 6000 interactions with about 3900 ligands. There is an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes almost 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at . G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2023, and supersedes data presented in the 2021/22, 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate. | |
650 | 7 | a MEDICIN OCH HÄLSOVETENSKAPx Medicinska och farmaceutiska grundvetenskaperx Farmakologi och toxikologi0 (SwePub)301022 hsv//swe |
650 | 7 | a MEDICAL AND HEALTH SCIENCESx Basic Medicinex Pharmacology and Toxicology0 (SwePub)301022 hsv//eng |
700 | 1 | a Christopoulos, Arthuru Monash Univ, Monash Inst Pharmaceut Sci, Parkville, Vic 3052, Australia.;Monash Univ, Dept Pharmacol, Parkville, Vic 3052, Australia.4 aut |
700 | 1 | a Davenport, Anthony P.u Univ Cambridge, Clin Pharmacol Unit, Cambridge CB2 0QQ, England.4 aut |
700 | 1 | a Kelly, Eamonnu Univ Bristol, Sch Physiol Pharmacol & Neurosci, Bristol BS8 1TD, Avon, England.4 aut |
700 | 1 | a Mathie, Alistair A.u Univ Suffolk, Sch EAST Engn Arts Sci & Technol, Ipswich IP4 1QJ, Suffolk, England.,Florida Int Univ, Miami, FL 33199 USA.4 aut |
700 | 1 | a Peters, John A.u Univ Dundee, Ninewells Hosp & Med Sch, Med Educ Inst, Neurosci Div, Dundee DD1 9SY, Angus, Scotland.4 aut |
700 | 1 | a Veale, Emma L.u Univ Greenwich, Medway Sch Pharm, Anson Bldg,Cent Ave, Chatham ME4 4TB, Kent, England.;Univ Kent, Medway, Anson Bldg,Cent Ave, Chatham ME4 4TB, Kent, England.4 aut |
700 | 1 | a Armstrong, Jane F.u Univ Edinburgh, Ctr Discovery Brain Sci, Edinburgh EH8 9XD, Midlothian, Scotland.4 aut |
700 | 1 | a Faccenda, Elenau Univ Edinburgh, Ctr Discovery Brain Sci, Edinburgh EH8 9XD, Midlothian, Scotland.4 aut |
700 | 1 | a Harding, Simon D.u Univ Edinburgh, Ctr Discovery Brain Sci, Edinburgh EH8 9XD, Midlothian, Scotland.4 aut |
700 | 1 | a Davies, Jamie A.u Univ Edinburgh, Ctr Discovery Brain Sci, Edinburgh EH8 9XD, Midlothian, Scotland.4 aut |
700 | 1 | a Abbracchio, Maria Piau Univ Milan, Milan, Italy.4 aut |
700 | 1 | a Abraham, Georgeu Univ Cambridge, Clin Pharmacol Unit, Cambridge CB2 0QQ, England.4 aut |
700 | 1 | a Agoulnik, Alexanderu NIH, Bldg 10, Bethesda, MD 20892 USA.,Univ Bristol, Sch Physiol Pharmacol & Neurosci, Bristol BS8 1TD, Avon, England.,Univ Nottingham, Med Sch, Sch Life Sci, Nottingham NG7 2UH, England.4 aut |
700 | 1 | a Alexander, Wayneu Emory Univ, Atlanta, GA 30322 USA.4 aut |
700 | 1 | a Al-hosaini, Khaledu King Saud Univ, Riyadh, Saudi Arabia.4 aut |
700 | 1 | a Baeck, Magnusu Karolinska Institutet4 aut |
700 | 1 | a Baker, Jillian G.u Univ Nottingham, Med Sch, Sch Life Sci, Nottingham NG7 2UH, England.4 aut |
700 | 1 | a Barnes, Nicholas M.u Univ Birmingham, Birmingham, Warwickshire, England.4 aut |
700 | 1 | a Bathgate, Rossu Florey Inst Neurosci & Mental Hlth, Melbourne, Vic, Australia.4 aut |
700 | 1 | a Beaulieu, Jean-Martinu Univ Toronto, Toronto, ON, Canada.4 aut |
700 | 1 | a Beck-Sickinger, Annette G.u Univ Leipzig, Leipzig, Germany.4 aut |
700 | 1 | a Behrens, Maiku Tech Univ Munich, Freising Weihenstephan, Germany.4 aut |
700 | 1 | a Bernstein, Kenneth E.u Cedars Sinai Med Ctr, Los Angeles, CA 90048 USA.,Univ Sherbrooke, Sherbrooke, PQ, Canada.4 aut |
700 | 1 | a Bettler, Bernhardu Univ Basel, Basel, Switzerland.,Univ Leicester, Leicester, Leics, England.4 aut |
700 | 1 | a Birdsall, Nigel J. M.u Francis Crick Inst, London, England.,Univ Cambridge, Clin Pharmacol Unit, Cambridge CB2 0QQ, England.,French Natl Ctr Sci Res CNRS, Valbonne, France.4 aut |
700 | 1 | a Blaho, Victoriau Sanford Burnham Prebys Med Discovery Inst, La Jolla, CA USA.4 aut |
700 | 1 | a Boulay, Francoisu Univ Grenoble Alpes, Grenoble, France.4 aut |
700 | 1 | a Bousquet, Corinneu French Inst Hlth & Med Res INSERM, Toulouse, France.4 aut |
700 | 1 | a Braeuner-Osborne, Hansu Univ Copenhagen, Copenhagen, Denmark.4 aut |
700 | 1 | a Burnstock, Geoffreyu UCL, London, England.4 aut |
700 | 1 | a Calo, Girolamou Univ Padua, Padua, Italy.4 aut |
700 | 1 | a Castano, Justo P.u Univ Cordoba, Cordoba, Spain.4 aut |
700 | 1 | a Catt, Kevin J.u NIH, Bldg 10, Bethesda, MD 20892 USA.4 aut |
700 | 1 | a Ceruti, Stefaniau Univ Milan, Milan, Italy.4 aut |
700 | 1 | a Chazot, Paulu Univ Durham, Durham, England.4 aut |
700 | 1 | a Chiang, Nanu Harvard Univ, Boston, MA 02115 USA.4 aut |
700 | 1 | a Chini, Biceu Univ Milano Bicocca, Vedano Al Lambro, Italy.4 aut |
700 | 1 | a Chun, Jeroldu Univ Calif San Diego, La Jolla, CA 92093 USA.4 aut |
700 | 1 | a Cianciulli, Antoniau Univ Bari, Bari, Italy.4 aut |
700 | 1 | a Civelli, Olivieru Univ Calif Irvine, Irvine, CA USA.4 aut |
700 | 1 | a Clapp, Lucie H.u UCL, London, England.4 aut |
700 | 1 | a Couture, Rejeanu Univ Montreal, Montreal, PQ, Canada.4 aut |
700 | 1 | a Cox, Helen M.u Kings Coll London, London, England.4 aut |
700 | 1 | a Csaba, Zsoltu French Inst Hlth & Med Res INSERM, Paris, France.4 aut |
700 | 1 | a Dahlgren, Claes,d 1949u Gothenburg University,Göteborgs universitet,Institutionen för medicin, avdelningen för reumatologi och inflammationsforskning,Institute of Medicine, Department of Rheumatology and Inflammation Research,Univ Gothenburg, Gothenburg, Sweden.4 aut0 (Swepub:gu)xdahcl |
700 | 1 | a Dent, Gordonu Keele Univ, Keele, Staffs, England.4 aut |
700 | 1 | a Douglas, Steven D.u Univ Penn, Philadelphia, PA 19104 USA.4 aut |
700 | 1 | a Dournaud, Pascalu French Inst Hlth & Med Res INSERM, Paris, France.4 aut |
700 | 1 | a Eguchi, Satoruu Temple Univ, Philadelphia, PA 19122 USA.4 aut |
700 | 1 | a Escher, Emanuelu Boston Univ, Boston, MA 02215 USA.,Univ Bonn, Bonn, Germany.4 aut |
700 | 1 | a Filardo, Edward J.u Univ Iowa, Iowa City, IA USA.4 aut |
700 | 1 | a Fong, Tungu Labcorp Drug Dev, Somerset, NJ USA.4 aut |
700 | 1 | a Fumagalli, Martau Univ Milan, Milan, Italy.4 aut |
700 | 1 | a Gainetdinov, Raul R.u St Petersburg State Univ, St Petersburg, Russia.,Univ Calgary, Calgary, AB, Canada.4 aut |
700 | 1 | a Garelja, Michael L.u Univ Otago, Dunedin, New Zealand.4 aut |
700 | 1 | a de Gasparo, Marcu MG Consulting Co, Basel, Switzerland.4 aut |
700 | 1 | a Gerard, Craigu Harvard Univ, Boston, MA 02115 USA.4 aut |
700 | 1 | a Gershengorn, Marvinu NIH, Bldg 10, Bethesda, MD 20892 USA.4 aut |
700 | 1 | a Gobeil, Fernandu Univ Sherbrooke, Sherbrooke, PQ, Canada.4 aut |
700 | 1 | a Goodfriend, Theodore L.u Univ Wisconsin, Madison, WI USA.4 aut |
700 | 1 | a Goudet, Cyrilu French Natl Ctr Sci Res, Montpellier, France.4 aut |
700 | 1 | a Graetz, Lukasu Karolinska Institutet4 aut |
700 | 1 | a Gregory, Karen J.u Monash Univ, Monash Inst Pharmaceut Sci, Parkville, Vic 3052, Australia.;Monash Univ, Dept Pharmacol, Parkville, Vic 3052, Australia.4 aut |
700 | 1 | a Gundlach, Andrew L.u Florey Inst Neurosci & Mental Hlth, Melbourne, Vic, Australia.4 aut |
700 | 1 | a Hamann, Joergu Univ Amsterdam, Amsterdam, Netherlands.4 aut |
700 | 1 | a Hanson, Julienu Univ Liege, Liege, Belgium.4 aut |
700 | 1 | a Hauger, Richard L.u Univ Calif San Diego, La Jolla, CA 92093 USA.4 aut |
700 | 1 | a Hay, Debbie L.u Univ Otago, Dunedin, New Zealand.4 aut |
700 | 1 | a Heinemann, Akosu Med Univ Graz, Graz, Austria.4 aut |
700 | 1 | a Herr, Deronu San Diego State Univ, San Diego, CA 92182 USA.4 aut |
700 | 1 | a Hollenberg, Morley D.u Univ Calgary, Calgary, AB, Canada.4 aut |
700 | 1 | a Holliday, Nicholas D.u Univ Nottingham, Med Sch, Sch Life Sci, Nottingham NG7 2UH, England.4 aut |
700 | 1 | a Horiuchi, Mastguguu Ehime Univ, Matsuyama, Ehime, Japan.4 aut |
700 | 1 | a Hoyer, Danielu Univ Melbourne, Melbourne, Vic, Australia.4 aut |
700 | 1 | a Hunyady, Laszlou Semmelwe Univ, Budapest, Hungary.4 aut |
700 | 1 | a Husain, Ahsanu Emory Univ, Atlanta, GA 30322 USA.4 aut |
700 | 1 | a Ijzerman, Adriaan P.u Leiden Univ, Leiden, Netherlands.4 aut |
700 | 1 | a Inagami, Tadashiu Vanderbilt Univ, 221 Kirkland Hall, Nashville, TN 37235 USA.4 aut |
700 | 1 | a Jacobson, Kenneth A.4 aut |
700 | 1 | a Jensen, Robert T.u NIH, Bldg 10, Bethesda, MD 20892 USA.4 aut |
700 | 1 | a Jockers, Ralfu French Inst Hlth & Med Res INSERM, Paris, France.4 aut |
700 | 1 | a Jonnalagadda, Deepau Sanford Burnham Prebys Med Discovery Inst, La Jolla, CA USA.4 aut |
700 | 1 | a Karnik, Sadashivau Lerner Res Inst, Cleveland, OH USA.4 aut |
700 | 1 | a Kaupmann, Klemensu Novartis, Basel, Switzerland.,Friedrich Schiller Univ Jena, Jena, Germany.4 aut |
700 | 1 | a Kemp, Jacquelineu Cleveland Clin, Lerner Res Inst, Cleveland, OH 44106 USA.4 aut |
700 | 1 | a Kennedy, Charlesu Strathclyde Univ, Glasgow, Lanark, Scotland.4 aut |
700 | 1 | a Kihara, Yasuyukiu Sanford Burnham Prebys Med Discovery Inst, La Jolla, CA USA.4 aut |
700 | 1 | a Kitazawa, Takiou Rakuno Gakuen Univ, Ebetsu, Hokkaido, Japan.4 aut |
700 | 1 | a Kozielewicz, Pawelu Karolinska Institutet4 aut |
700 | 1 | a Kreienkamp, Hans-Juergenu Univ Hamburg, Hamburg, Germany.4 aut |
700 | 1 | a Kukkonen, Jyrki P.u Univ Helsinki, Helsinki, Finland.4 aut |
700 | 1 | a Langenhan, Tobiasu Univ Leipzig, Leipzig, Germany.4 aut |
700 | 1 | a Larhammar, Dan,d 1956-u Uppsala universitet,Forskargrupp Dan Larhammar,Science for Life Laboratory, SciLifeLab4 aut0 (Swepub:uu)dla05000 |
700 | 1 | a Leach, Katieu Monash Univ, Monash Inst Pharmaceut Sci, Parkville, Vic 3052, Australia.;Monash Univ, Dept Pharmacol, Parkville, Vic 3052, Australia.4 aut |
700 | 1 | a Lecca, Davideu Univ Milan, Milan, Italy.4 aut |
700 | 1 | a Lee, John D.u Univ Queensland, Brisbane, Qld, Australia.4 aut |
700 | 1 | a Leeman, Susan E.4 aut |
700 | 1 | a Leprince, Jeromeu Univ Rouen, Rouen, France.,Mayo Fdn Med Educ & Res, Scottsdale, AZ USA.4 aut |
700 | 1 | a Li, Xaria X.u Univ Queensland, Toowoomba, Qld, Australia.4 aut |
700 | 1 | a Lolait, Stephen J.u Univ Bristol, Sch Physiol Pharmacol & Neurosci, Bristol BS8 1TD, Avon, England.4 aut |
700 | 1 | a Lupp, Amelieu Friedrich Schiller Univ Jena, Jena, Germany.4 aut |
700 | 1 | a Macrae, Robynu Univ Cambridge, Cambridge, England.4 aut |
700 | 1 | a Maguire, Janet4 aut |
700 | 1 | a Malfacini, Davideu Univ Padua, Padua, Italy.4 aut |
700 | 1 | a Mazella, Jean4 aut |
700 | 1 | a Mcardle, Craig A.4 aut |
700 | 1 | a Melmed, Shlomou Cedars Sinai Med Ctr, Los Angeles, CA 90048 USA.4 aut |
700 | 1 | a Michel, Martin C.u Johannes Gutenberg Univ Mainz, Mainz, Germany.,Deakin Univ, Waurn Ponds, Australia.4 aut |
700 | 1 | a Miller, Laurence J.4 aut |
700 | 1 | a Mitolo, Vincenzou Univ Bari, Bari, Italy.4 aut |
700 | 1 | a Mouillac, Bernardu French Natl Ctr Sci Res, Montpellier, France.4 aut |
700 | 1 | a Mueller, Christa E.4 aut |
700 | 1 | a Murphy, Philip M.u Edge Hill Univ, Bethesda, MD USA.4 aut |
700 | 1 | a Nahon, Jean-Louisu French Natl Ctr Sci Res CNRS, Valbonne, France.4 aut |
700 | 1 | a Ngo, Tonyu Sanford Burnham Prebys Med Discovery Inst, La Jolla, CA USA.4 aut |
700 | 1 | a Norel, Xavieru French Inst Hlth & Med Res INSERM, Paris, France.4 aut |
700 | 1 | a Nyimanu, Duuameneu Univ Cambridge, Cambridge, England.4 aut |
700 | 1 | a O'Carroll, Anne-Marieu Univ Bristol, Sch Physiol Pharmacol & Neurosci, Bristol BS8 1TD, Avon, England.4 aut |
700 | 1 | a Offermanns, Stefanu Max Planck Inst Heart & Lung Res, Bad Nauheim, Germany.4 aut |
700 | 1 | a Panaro, Maria Antoniettau Univ Bari, Bari, Italy.4 aut |
700 | 1 | a Parmentier, Marcu Free Univ Brussels, Brussels, Belgium.4 aut |
700 | 1 | a Pertwee, Roger G.u Univ Aberdeen, Aberdeen, Scotland.4 aut |
700 | 1 | a Pin, Jean-Philippeu Univ Montpellier, Montpellier, France.4 aut |
700 | 1 | a Prossnitz, Eric R.u Univ New Mexico, Albuquerque, NM 87131 USA.4 aut |
700 | 1 | a Quinn, Marku Montana State Univ, Bozeman, MT 59717 USA.4 aut |
700 | 1 | a Ramachandran, Rithwik4 aut |
700 | 1 | a Ray, Manishau Sanford Burnham Prebys Med Discovery Inst, La Jolla, CA USA.4 aut |
700 | 1 | a Reinscheid, Rainer K.4 aut |
700 | 1 | a Rondard, Philippeu Univ Montpellier, Montpellier, France.4 aut |
700 | 1 | a Rovati, G. Enricou Univ Milan, Milan, Italy.4 aut |
700 | 1 | a Ruzza, Chiarau Univ Ferrara, Ferrara, Italy.4 aut |
700 | 1 | a Sanger, Gareth J.u Queen Mary Univ London, London, England.4 aut |
700 | 1 | a Schoeneberg, Torstenu Univ Leipzig, Leipzig, Germany.4 aut |
700 | 1 | a Schulte, Gunnaru Karolinska Institutet4 aut |
700 | 1 | a Schulz, Stefanu Friedrich Schiller Univ Jena, Jena, Germany.,Univ Auckland, Auckland, New Zealand.4 aut |
700 | 1 | a Segaloff, Deborah L.u Univ Iowa, Iowa City, IA USA.4 aut |
700 | 1 | a Serhan, Charles N.u Harvard Univ, Boston, MA 02115 USA.4 aut |
700 | 1 | a Singh, Khuraijam Dhanachandrau Cleveland Clin, Lerner Res Inst, Cleveland, OH 44106 USA.4 aut |
700 | 1 | a Smith, Craig M.4 aut |
700 | 1 | a Stoddart, Leigh A.4 aut |
700 | 1 | a Sugimoto, Yukihikou Kumamoto Univ, Kumamoto, Japan.4 aut |
700 | 1 | a Summers, Rogeru Monash Univ, Melbourne, Vic, Australia.4 aut |
700 | 1 | a Tan, Valerie P.u Univ Calif San Diego, La Jolla, CA 92093 USA.4 aut |
700 | 1 | a Thal, Davidu Monash Univ, Melbourne, Vic, Australia.4 aut |
700 | 1 | a Thomas, Walter ( Wally)u Univ Queensland, Toowoomba, Qld, Australia.4 aut |
700 | 1 | a Timmermans, Pieter B. M. W. M.4 aut |
700 | 1 | a Tirupula, Kalyanu Cleveland Clin, Lerner Res Inst, Cleveland, OH 44106 USA.4 aut |
700 | 1 | a Toll, Lawrenceu Florida Atlantic Univ, Jupiter, FL USA.4 aut |
700 | 1 | a Tulipano, Giovanniu Univ Brescia, Brescia, Italy.4 aut |
700 | 1 | a Unal, Hamiyetu Cleveland Clin, Cleveland, OH 44106 USA.4 aut |
700 | 1 | a Unger, Thomasu Maastricht Univ, Maastricht, Netherlands.4 aut |
700 | 1 | a Valant, Celineu Monash Univ, Melbourne, Vic, Australia.4 aut |
700 | 1 | a Vanderheyden, Patricku Free Univ Brussels, Brussels, Belgium.4 aut |
700 | 1 | a Vaudry, Davidu Univ Rouen, Rouen, France.4 aut |
700 | 1 | a Vaudry, Hubertu Univ Rouen, Rouen, France.4 aut |
700 | 1 | a Vilardaga, Jean-Pierreu Univ Pittsburgh, Pittsburgh, PA USA.4 aut |
700 | 1 | a Walker, Christopher S.4 aut |
700 | 1 | a Wang, Ji Mingu NCI, Frederick, MD 21701 USA.4 aut |
700 | 1 | a Ward, Donald T.u Univ Manchester, Manchester, Lancs, England.4 aut |
700 | 1 | a Wester, Hans-Juergenu Tech Univ Munich, Munich, Germany.4 aut |
700 | 1 | a Willars, Gary B.4 aut |
700 | 1 | a Williams, Tom Lloydu Univ Cambridge, Cambridge, England.4 aut |
700 | 1 | a Woodruff, Trent M.u Univ Queensland, Toowoomba, Qld, Australia.4 aut |
700 | 1 | a Yao, Chengcanu Univ Edinburgh, Edinburgh, Midlothian, Scotland.4 aut |
700 | 1 | a Ye, Richard D.u Chinese Univ Hong Kong, Shenzhen, Hong Kong, Peoples R China.4 aut |
710 | 2 | a Univ Nottingham, Med Sch, Sch Life Sci, Nottingham NG7 2UH, England.b Monash Univ, Monash Inst Pharmaceut Sci, Parkville, Vic 3052, Australia.;Monash Univ, Dept Pharmacol, Parkville, Vic 3052, Australia.4 org |
773 | 0 | t BRITISH JOURNAL OF PHARMACOLOGYd : British pharmacological societyg 180q 180x 0007-1188x 1476-5381 |
856 | 4 | u https://doi.org/10.1111/bph.16177y Fulltext |
856 | 4 | u https://uu.diva-portal.org/smash/get/diva2:1834555/FULLTEXT01.pdfx primaryx Raw objecty fulltext:print |
856 | 4 8 | u https://gup.ub.gu.se/publication/334432 |
856 | 4 8 | u https://doi.org/10.1111/bph.16177 |
856 | 4 8 | u https://urn.kb.se/resolve?urn=urn:nbn:se:uu:diva-521895 |
856 | 4 8 | u http://kipublications.ki.se/Default.aspx?queryparsed=id:154895192 |
856 | 4 8 | u http://kipublications.ki.se/Default.aspx?queryparsed=id:154633669 |
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